Lersivirine: a Non-Nucleoside Reverse Transcriptase Inhibitor with Activity against Drug-Resistant Human Immunodeficiency Virus-1.

Abstract:

The non-nucleoside reverse transcriptase inhibitors (NNRTIs) are key ...

Polymerases:

Topics:

Mutational Analysis, Structure and Structure/Function, Reverse Transcriptase

Status:

new topics/pols set partial results complete validated

Results:

Polymerase Reference Property Result Context
HIV RT Lersivirine: a Non-Nucleoside Reverse Transcriptase Inhibitor with Activity against Drug-Resistant Human Immunodeficiency Virus-1. Reverse Transcriptase Activity Yes
HIV RT K103N Lersivirine: a Non-Nucleoside Reverse Transcriptase Inhibitor with Activity against Drug-Resistant Human Immunodeficiency Virus-1. Reverse Transcriptase Activity Yes

Structures:

2WON 2WOM