Design of annulated pyrazoles as inhibitors of HIV-1 reverse transcriptase.
Sweeney ZK, Harris SF, Arora SF, Javanbakht H, Li Y, Fretland J, Davidson JP, Billedeau JR, Gleason SK, Hirschfeld DR, Kennedy-Smith JJ, Mirzadegan T, Roetz R, Smith M, Sperry S, Suh JM, Wu J, Tsing S, VillaseƱor AG, Paul A, Su G, Heilek GM, Hang JQ, Zhou AS, Jernelius JA, Zhang FJ, Klumpp K
J Med Chem (2008), Volume 51, Page 7449
Abstract:
Polymerases:
Topics:
Reverse Transcriptase
Status:
new | topics/pols set | partial results | complete | validated |
Results:
Polymerase | Reference | Property | Result | Context |
---|---|---|---|---|
HIV RT | Design of annulated pyrazoles as inhibitors of HIV-1 reverse transcriptase. | Reverse Transcriptase Activity | Yes |