N1-Alkyl pyrimidinediones as non-nucleoside inhibitors of HIV-1 reverse transcriptase.

Abstract:

A series of N1-alkyl pyrimidinediones were designed, synthesized and ...

Polymerases:

Topics:

Structure and Structure/Function, Reverse Transcriptase

Status:

new topics/pols set partial results complete validated

Results:

Polymerase Reference Property Result Context
HIV RT N1-Alkyl pyrimidinediones as non-nucleoside inhibitors of HIV-1 reverse transcriptase. Reverse Transcriptase Activity Yes

Entry validated by:

Structures:

3LAN 3LAM 3LAL